SCHEMBL28115405

SCHEMBL28115405

CN(Cc1ccccc1)C1C[C@H]2CC(=O)C[C@H]2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.50
JAK1 P23458 1/20 0.50
NAAA Q02083 2/20 0.45
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
GRIN2B Q13224 1/20 0.43
SLC18A3 Q16572 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
AGTR2 P50052 2/20 0.41
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
AOC3 Q16853 1/20 0.39
LMNA P02545 1/20 0.39
MAOA P21397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28115404 1.00 JAK2 (0.50) JAK2JAK1NAAADDB1CRBN
SCHEMBL21595465 0.83 YTHDC1 (0.44) JAK2JAK1DDB1CRBNGRIN2B
SCHEMBL21595464 0.83 YTHDC1 (0.44) JAK2JAK1DDB1CRBNGRIN2B
SCHEMBL15077587 0.83 DDB1 (0.45) JAK2JAK1NAAADDB1CRBN
SCHEMBL15077588 0.82 JAK2 (0.52) JAK2JAK1NAAADDB1CRBN
SCHEMBL23950410 0.80 NAAA (0.49) JAK2JAK1NAAADDB1CRBN
SCHEMBL31715951 0.80 NAAA (0.49) JAK2JAK1NAAADDB1CRBN
SCHEMBL10039726 0.79 NAAA (0.46) JAK2JAK1NAAADDB1CRBN
SCHEMBL28115401 0.79 SLC18A3 (0.50) JAK2JAK1NAAADDB1CRBN
SCHEMBL28115399 0.79 SLC18A3 (0.50) JAK2JAK1NAAADDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106336406-B Having beta2Octahydropentalene derivatives with receptor agonistic and M receptor antagonistic activity and their medical use 四川海思科制药有限公司 2020-01-03 CN disclosed
CN-106336406-A Octahydrocyclopentadiene derivative with beta2 receptor agonisis and M receptor antagonism activity, and use thereof in medicines 四川海思科制药有限公司 2017-01-18 CN disclosed