SCHEMBL28116469

SCHEMBL28116469

O=Cc1cccc(OC(F)(F)F)c1Oc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.56
KMT2A Q03164 2/20 0.56
GAA P10253 1/20 0.56
ALDH1A1 P00352 5/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HPGD P15428 2/20 0.41
HTT P42858 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TSHR P16473 1/20 0.37
TLR2 O60603 2/20 0.37
TLR4 O00206 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
PTGES2 Q9H7Z7 1/20 0.36
SRC P12931 2/20 0.36
MEN1 O00255 1/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16470387 0.84 SRC (0.41) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL27645264 0.82 ALDH1A1 (0.39) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL18112650 0.80 CA1 (0.53) LMNAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL96815 0.78 ALDH1A1 (0.55) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL31241188 0.78 LMNA (0.50) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL28195278 0.78 LMNA (0.50) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL6955863 0.76 LMNA (0.60) LMNAKMT2AGAAALDH1A1CYP1A2
SCHEMBL9590947 0.76 CTNNB1 (0.45) GAAALDH1A1HTTTDP1L3MBTL1
SCHEMBL5919466 0.76 SLC22A12 (0.42) PTGDR2PTGES2CA1CA2
SCHEMBL1252353 0.76 ALDH1A1 (0.42) LMNAGAAALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255679-B As NAThe heterocyclic compound and application thereof of V channel inhibitor 默克专利有限公司 2019-09-06 CN disclosed
CN-106255679-A As Naheterocyclic compound of V channel inhibitor and application thereof 默克专利有限公司 2016-12-21 CN disclosed