SCHEMBL28116653

SCHEMBL28116653

CC(C)c1ccc2nc(-c3cc(O)c(O)c(O)c3)[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
SCN10A Q9Y5Y9 1/20 0.50
AMY1A P0DUB6 3/20 0.47
MAPT P10636 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
TP53 P04637 2/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
ALDH1A1 P00352 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
GAA P10253 2/20 0.44
KDM4E B2RXH2 2/20 0.44
GLA P06280 2/20 0.44
RECQL P46063 2/20 0.44
RXFP1 Q9HBX9 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13160197 0.83 HDAC3 (0.65) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12763751 0.81 MAPT (0.62) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL28116651 0.81 NPC1 (0.63) AMY1AMAPTSMN1; SMN2TP53ALDH1A1
SCHEMBL28116665 0.77 ALDH1A1 (0.58) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL15945341 0.77 SCN10A (0.59) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12763752 0.76 NPC1 (0.67) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL27983509 0.75 ALDH1A1 (0.63) HDAC6MAPTSMN1; SMN2TP53MEN1
SCHEMBL13183515 0.74 NPC1 (0.66) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL9925390 0.72 HDAC3 (0.60) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL25521792 0.72 SMN1; SMN2 (0.55) HDAC6MAPTSMN1; SMN2TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104072425-B Benzimidazole compound and application thereof 大连理工大学 2016-12-07 CN claimed
CN-104072425-B Benzimidazole compound and application thereof 大连理工大学 2016-12-07 CN disclosed