SCHEMBL28119602

SCHEMBL28119602

COc1ccc(N(C)C(=O)C(Cc2ccccc2)OC(N)=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.53
PPARA Q07869 3/20 0.53
MAPK1 P28482 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
ATM Q13315 1/20 0.43
LDHA P00338 1/20 0.43
ACHE P22303 1/20 0.42
CIT O14578 1/20 0.41
RNF4 P78317 1/20 0.41
FPR2 P25090 1/20 0.41
ALDH1A1 P00352 2/20 0.41
SRR Q9GZT4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28711821 1.00 PPARG (0.53) PPARGPPARAMAPK1OPRM1OPRD1
SCHEMBL28838109 0.90 SRR (0.46) PPARGPPARACITALDH1A1SRR
SCHEMBL28119856 0.88 PDK1 (0.46) PPARGPPARAATMALDH1A1
SCHEMBL28119599 0.87 PARP15 (0.44) PPARGPPARAALDH1A1
SCHEMBL28119870 0.86 RNF4 (0.53) PPARGPPARAMAPK1RNF4ALDH1A1
SCHEMBL28119603 0.85 L3MBTL1 (0.42) PPARGPPARAMAPK1ALDH1A1
SCHEMBL28732592 0.85 HSP90AA1 (0.39) PPARGPPARALDHAALDH1A1
SCHEMBL28732594 0.85 HSP90AA1 (0.39) PPARGPPARALDHAALDH1A1
SCHEMBL28838104 0.84 PPARG (0.37) PPARGPPARAALDH1A1
SCHEMBL28753334 0.83 SCN9A (0.51) PPARGPPARAMAPK1LDHAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109836477-B Phenylalanine derivative containing benzothiadiazine-3-ketone 1, 1-dioxide and preparation method and application thereof 山东大学 2022-07-12 CN disclosed
CN-109897088-B Phenylalanine derivative containing N- (2-oxoethyl) benzene sulfonamide and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-109796418-B Phenylalanine derivative containing 4-phenyl-1, 2, 3-triazole and preparation method and application thereof 山东大学 2022-03-25 CN disclosed
CN-109824756-B Phenylalanine derivative containing 4- (benzenesulfonyl) piperazine-2-ketone and preparation method and application thereof 山东大学 2022-03-22 CN disclosed
CN-106458940-A Inhibitors of human immunodeficiency virus replication 百时美施贵宝公司 2017-02-22 CN disclosed