SCHEMBL28130528

SCHEMBL28130528

c1ccc(Oc2ccc(Oc3cncnc3)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 7/20 0.57
TSHR P16473 1/20 0.57
NR1H2 P55055 1/20 0.50
BAX Q07812 1/20 0.50
MAOA P21397 1/20 0.50
SOS1 Q07889 1/20 0.47
ATM Q13315 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CYP19A1 P11511 1/20 0.44
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
GSTP1 P09211 1/20 0.42
CA9 Q16790 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PLA2G2A P14555 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24710880 0.98 LTA4H (0.60) LTA4HTSHRNR1H2BAXMAOA
Diphenylether SCHEMBL28210066 0.85 LTA4H (0.71) LTA4HTSHRNR1H2BAXMAOA
SCHEMBL7017341 0.85 ATM (0.64) LTA4HTSHRNR1H2BAXMAOA
SCHEMBL9242002 0.82 LMNA (0.39) ATMLMNATDP1
SCHEMBL168543 0.81 LMNA (0.55) MAOACA1CA2LMNACA9
Diphenylether SCHEMBL27916363 0.80 LTA4H (0.63) LTA4HTSHRNR1H2BAXMAOA
SCHEMBL11396596 0.79 LTA4H (0.54) LTA4HCYP11B1CYP11B2CA1CA2
SCHEMBL8737455 0.79 TEAD4 (0.52) ATMCYP19A1TDP1SCN5ASCN9A
SCHEMBL178154 0.79 ALDH1A1 (0.64) TSHRMAOATDP1PARP10
SCHEMBL27761280 0.79 SOS1 (0.48) SOS1CA1CA2CYP19A1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103814016-B Compositions and methods for producing pyrimidine and pyridine compounds having BTK inhibitory activity 默克专利有限公司 2017-03-08 CN disclosed