SCHEMBL28131997

SCHEMBL28131997

CCCCS(=O)(=O)c1cccc(-c2ccncc2)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.48
LARS1 Q9P2J5 1/20 0.45
LRRK2 Q5S007 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
PRMT6 Q96LA8 1/20 0.41
CYP2D6 P10635 2/20 0.41
PRKCI P41743 1/20 0.41
KIF11 P52732 1/20 0.41
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
KDR P35968 1/20 0.40
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17364170 0.91 LARS1 (0.46) HTR6LARS1LRRK2CYP3A4CYP2C9
SCHEMBL2704870 0.88 CYP2C9 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8920560 0.86 CYP2C9 (0.45) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL2703373 0.83 CYP2C9 (0.48) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8745144 0.82 HDAC1 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL4630948 0.82 CYP2C9 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL14426918 0.79 NPC1 (0.50) HTR6CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL1228349 0.78 CYP2C9 (0.58) HTR6LARS1CYP3A4CYP2C9CYP2C19
SCHEMBL29297465 0.76 L3MBTL1 (0.50) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL30690007 0.76 ALOX5 (0.53) LARS1LRRK2KIF11NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113511997-A Pridopidine analogues, their preparation and use 普丽莱尼亚神经治疗有限公司 2021-10-19 CN claimed
CN-113511997-A Pridopidine analogues, their preparation and use 普丽莱尼亚神经治疗有限公司 2021-10-19 CN disclosed
CN-106456618-A Pridopidine analogues, their preparation and use 泰华制药工业有限公司 2017-02-22 CN disclosed