SCHEMBL28134397

SCHEMBL28134397

[CH2]c1cccc(-c2c(C)cc(N)cc2C)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.41
HTR7 P34969 1/20 0.38
SRC P12931 2/20 0.37
ALDH1A1 P00352 2/20 0.35
GRIA1 P42261 2/20 0.35
CACNG8 Q8WXS5 2/20 0.35
RPS6KA3 P51812 1/20 0.35
CYP3A4 P08684 2/20 0.33
MAOA P21397 1/20 0.33
TSHR P16473 1/20 0.33
PIK3CA P42336 1/20 0.33
FFAR1 O14842 1/20 0.33
IKBKE Q14164 1/20 0.33
IKBKB O14920 1/20 0.33
PDE10A Q9Y233 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2090907 0.88 HTR7 (0.46) MAP4K4HTR7SRCGRIA1CACNG8
SCHEMBL2093499 0.84 FFAR1 (0.36) MAP4K4HTR7SRCALDH1A1GRIA1
SCHEMBL16429717 0.77 RPS6KA3 (0.47) ALDH1A1RPS6KA3CYP3A4MAOATSHR
SCHEMBL8954027 0.74 ALDH1A1 (0.48) SRCALDH1A1GRIA1CACNG8RPS6KA3
SCHEMBL16431919 0.73 MAP4K4 (0.56) MAP4K4HTR7SRCALDH1A1GRIA1
SCHEMBL29557215 0.72 MAP4K4 (0.51) MAP4K4ALDH1A1CYP3A4MAOATSHR
SCHEMBL21539290 0.72 MAP4K4 (0.51) MAP4K4ALDH1A1CYP3A4MAOATSHR
SCHEMBL9848294 0.72 RAB9A (0.44) MAP4K4ALDH1A1
SCHEMBL12565770 0.71 HTR7 (0.53) MAP4K4HTR7SRCALDH1A1GRIA1
SCHEMBL28441441 0.70 ALDH1A1 (0.50) ALDH1A1CYP3A4TSHRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104592211-B Biphenyl compound and application thereof 广东东阳光药业有限公司 2018-10-16 CN disclosed
CN-104193731-B A kind of urea substituted biphenyl class compound and combinations thereof and purposes 广东东阳光药业有限公司 2017-03-15 CN disclosed