SCHEMBL28136392

SCHEMBL28136392

Cc1ccccc1Cn1ccc(C(N)=O)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 1/20 0.51
CACNA1G O43497 2/20 0.50
CACNA1H O95180 2/20 0.50
CACNA1I Q9P0X4 2/20 0.50
LMNA P02545 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
POLB P06746 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15964805 0.82 NPC1 (0.48) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL4288842 0.78 HDAC1 (0.56) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL3440017 0.76 KMT2A (0.66) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL29049999 0.76 KMT2A (0.51) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL4726770 0.76 SMN1; SMN2 (0.50) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL29757100 0.75 KLKB1 (0.45) RAB9ALMNAKDM4EMAPTSMN1; SMN2
SCHEMBL22888044 0.75 KLKB1 (0.45) RAB9ALMNAKDM4EMAPTSMN1; SMN2
SCHEMBL15964729 0.75 PTGER1 (0.56) KDM4ETSHR
SCHEMBL15520038 0.74 LMNA (0.40) KMT2AMEN1NPC1RAB9ACACNA1G
SCHEMBL3439964 0.74 CACNA1G (0.64) KMT2AMEN1NPC1RAB9ACACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106573006-A Heterocyclic amides of RIP1 kinase inhibitors as pharmaceuticals 葛兰素史密斯克莱知识产权发展有限公司 2017-04-19 CN disclosed