SCHEMBL28138447

SCHEMBL28138447

NC(=O)C1Cc2cccc3cccc1c23

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.49
MTNR1B P49286 10/20 0.49
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
OPRL1 P41146 1/20 0.43
KDM4E B2RXH2 1/20 0.39
PARP1 P09874 3/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8440245 0.98 MTNR1A (0.48) MTNR1AMTNR1BOPRM1OPRD1OPRK1
Formic Acid SCHEMBL28598514 0.94 MTNR1A (0.45) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL28248972 0.89 MTNR1A (0.41) MTNR1AMTNR1BOPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL28260890 0.87 MTNR1A (0.40) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL9240061 0.86 MTNR1A (0.51) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL5380872 0.84 MTNR1A (0.50) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL30066901 0.84 MTNR1A (0.50) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL27343077 0.83 MTNR1A (0.48) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL28599443 0.83 MTNR1A (0.49) MTNR1AMTNR1BOPRM1OPRD1OPRK1
SCHEMBL5370015 0.83 MTNR1A (0.56) MTNR1AMTNR1BOPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN claimed
CN-108884106-A POLYCYCLIC COMPOUNDS AS INHIBITORS OF BRUTON'S TYROSINE KINASE 詹森药业有限公司 2018-11-23 CN claimed
CN-108794544-A It is used to prepare the alpha-nickel diimine compound of asymmetry containing nitro, intermediate, the Preparation method and use of ultra-high molecular weight polyethylene 中国科学院化学研究所 2018-11-13 CN claimed
CN-108794545-A It is used to prepare the alpha-nickel diimine compound of asymmetry containing tertiary butyl, the Preparation method and use of ultra-high molecular weight polyethylene elastomer 中国科学院化学研究所 2018-11-13 CN claimed
CN-106632506-A 4,4'-difluorobenzhydryl containing asymmetric alpha-diimine nickel complex, and intermediate, preparation method and application thereof 中国科学院化学研究所 2017-05-10 CN claimed
CN-113121562-B Polycyclic compounds as inhibitors of bruton's tyrosine kinase 詹森药业有限公司 2022-09-13 CN disclosed
CN-113105475-B Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2022-09-09 CN disclosed
CN-113121562-A Polycyclic compounds as inhibitors of bruton's tyrosine kinase 詹森药业有限公司 2021-07-16 CN disclosed
CN-113105475-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2021-07-13 CN disclosed
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN disclosed
CN-108884106-A POLYCYCLIC COMPOUNDS AS INHIBITORS OF BRUTON'S TYROSINE KINASE 詹森药业有限公司 2018-11-23 CN disclosed