SCHEMBL28142156

SCHEMBL28142156

CCCCCN(N)c1cccc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.41
LTB4R2 Q9NPC1 2/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
EPHX1 P07099 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
CETP P11597 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
IDO1 P14902 2/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7752962 0.81 AR (0.45) LTB4R2HDAC3HDAC1HDAC2HTR2A
SCHEMBL21169213 0.77 CETP (0.47) LTB4R2HTR2AHTR2CHTR2BTSHR
SCHEMBL253120 0.75 NPC1 (0.47)
SCHEMBL19265466 0.74 HTR7 (0.43) LTB4R2HTR2AHTR2CHTR2BTSHR
SCHEMBL5500471 0.74 CYP3A4 (0.44) LTB4R2HTR2AHTR2CHTR2BTSHR
SCHEMBL11265336 0.74 LTB4R2 (0.43) LTB4R2HDAC3HDAC1HDAC2EPHX1
SCHEMBL23072505 0.74 TAAR1 (0.46) HTR2AHTR2CHTR2BTSHRMAPK1
SCHEMBL8626864 0.73 CYP3A4 (0.55) HTR2AHTR2CHTR2BTSHRMAPK1
SCHEMBL6477185 0.73 NPC1 (0.50)
SCHEMBL6488829 0.73 NPC1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106660962-A Arylhydrazides containing 2-pyridone moieties for use as selective antibacterial agents ABAC治疗法有限公司 2017-05-10 CN claimed