SCHEMBL2814513

SCHEMBL2814513

c1ccc(CN2CCC3NNc4nc(NCc5cccc(-c6ccccc6)c5)nc2c43)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.37
ACHE P22303 4/20 0.36
BACE1 P56817 2/20 0.36
HTR5A P47898 1/20 0.36
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
TPH1 P17752 1/20 0.33
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
TNIK Q9UKE5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2812302 0.92 ACHE (0.37) ACHEBACE1HTR5AALDH1A1MEN1
SCHEMBL2811945 0.91 ACHE (0.38) ACHEBACE1ALDH1A1MEN1LMNA
SCHEMBL2812214 0.87 ADORA2A (0.42) ALDH1A1SMN1; SMN2KDM4EHSD17B10
SCHEMBL2808425 0.86 MRGPRX1 (0.39) HTR5AHRH2HRH1HRH4HRH3
SCHEMBL2810284 0.85 OGA (0.40)
SCHEMBL2816684 0.84 ACHE (0.47) ACHEBACE1LMNASMN1; SMN2CYP3A4
SCHEMBL2816411 0.84 ACHE (0.47) CXCR4ACHEBACE1ALDH1A1MEN1
SCHEMBL2812972 0.84 SIGMAR1 (0.38) ACHEBACE1MEN1KMT2AHRH1
SCHEMBL2814798 0.84 SIGMAR1 (0.40) ACHE
SCHEMBL537584 0.83 ACHE (0.45) ACHEBACE1MEN1KMT2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8343983-B2 Substituted pyrazolo-pyrimidine compounds ARQULE, INC. (US) 2013-01-01 US disclosed
US-20100249110-A1 SUBSTITUTED PYRAZOLO-PYRIMIDINE COMPOUNDS ARQULE, INC. (US) 2010-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100249110-A1 SUBSTITUTED PYRAZOLO-PYRIMIDINE COMPOUNDS DPYD, TYMP, TP53 CXCR4 492/4885ACHE 4402/4885BACE1 3588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.