Piperazine

Piperazine

SCHEMBL28145353

C1CNCCN1.Cc1ccnn1C

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.38
OXTR P30559 2/20 0.38
AVPR1A P37288 2/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPK1 P28482 1/20 0.35
SOD3 P08294 1/20 0.35
PLAT P00750 1/20 0.33
ADRB1 P08588 2/20 0.32
ADRB2 P07550 1/20 0.32
NCF1 P14598 1/20 0.32
PLD1 Q13393 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL28865391 0.88 MEN1 (0.39) COMTOXTRAVPR1ARAB9AALDH1A1
SCHEMBL257689 0.86
Pyridine SCHEMBL28065595 0.74 TSHR (0.39) COMTOXTRAVPR1ARAB9AALDH1A1
SCHEMBL16687146 0.70
SCHEMBL16692488 0.70
SCHEMBL23505274 0.69 PLD1 (0.46) ALDH1A1ADRB1ADRB2NCF1PLD1
SCHEMBL27516034 0.69 OXTR (0.45) OXTRAVPR1AALDH1A1MEN1MAPT
SCHEMBL2390106 0.69 RAB9A (0.35) COMTOXTRAVPR1ARAB9AALDH1A1
SCHEMBL15941963 0.68 PLAT (0.49) ALDH1A1MEN1MAPTPKMALOX15
SCHEMBL15950966 0.68 MEN1 (0.64) ALDH1A1MEN1MAPTPKMALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105929082-B A kind of method of Pyrazine and pyridine substance in separation determination saliva 云南中烟工业有限责任公司 2018-08-21 CN claimed
CN-106715518-B Conjugated polymer 默克专利有限公司 2019-10-25 CN disclosed
CN-109171004-A A kind of compounding maple extract Maillard reaction fragrance, preparation method and the application in papermaking-method reconstituted tobaccos 河南中烟工业有限责任公司 2019-01-11 CN disclosed
CN-108593814-A The quantitative detecting method of nitrogenous compound in a kind of white wine 北京工商大学 2018-09-28 CN disclosed
CN-105330821-B The copolymer of 2-glycidyl ether capped polysiloxane compound and non-aromatic polyamines 罗门哈斯电子材料有限公司 2018-08-28 CN disclosed
CN-107460106-A A kind of method of the content of alkyl pyrazine compound in raising vinegar 福建农林大学 2017-12-12 CN disclosed
CN-105353045-B The detection method of pyrazine compounds in a kind of Maotai-flavor liquor 贵州省产品质量监督检验院 2017-09-22 CN disclosed
CN-106715518-A Conjugated polymers 默克专利有限公司 2017-05-24 CN disclosed