SCHEMBL28146261

SCHEMBL28146261

O=[SH](=O)Cc1ccc(-c2cc(Cl)cnc2Br)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.34
PTGS2 P35354 15/20 0.34
PTGS1 P23219 8/20 0.34
ABCC4 O15439 1/20 0.33
ABCB11 O95342 1/20 0.33
PDE4D Q08499 1/20 0.33
MAPK14 Q16539 1/20 0.33
MAP4K4 O95819 1/20 0.32
KDR P35968 1/20 0.32
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28147339 0.82 FFAR4 (0.37) FFAR4PTGS2PTGS1ABCC4ABCB11
SCHEMBL27585000 0.76 PTGS2 (0.62) FFAR4PTGS2PTGS1ABCC4ABCB11
SCHEMBL24809552 0.74 JAK2 (0.50) PTGS2PTGS1MAP4K4KDR
SCHEMBL6069777 0.72 PTGS2 (0.63) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL27885060 0.71 FYN (0.43) MAP4K4
SCHEMBL27635241 0.69 CYP19A1 (0.38)
SCHEMBL27885058 0.69 HTT (0.41) MAP4K4
SCHEMBL14198821 0.67 IDO1 (0.46)
SCHEMBL28051403 0.67 USP7 (0.57) MAP4K4
SCHEMBL27459333 0.66 MAPK1 (0.52) FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106632002-A Preparation technology of etoricoxib and reference substance 5-chloro-3-(4-(methyl sulphonyl)phenyl)-2,3-bipyridine of etoricoxib 贵州大学 2017-05-10 CN disclosed