SCHEMBL28146262

SCHEMBL28146262

CS(=O)(=O)c1ccc(-c2cccnc2-c2cccnc2Cl)cc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.69
PTGS1 P23219 8/20 0.69
ABCC4 O15439 1/20 0.50
ABCB11 O95342 1/20 0.50
PDE4D Q08499 1/20 0.50
MAPK14 Q16539 1/20 0.50
PIP4K2A P48426 2/20 0.45
PIP4K2C Q8TBX8 2/20 0.45
PIP4K2B P78356 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170026 0.91 PTGS2 (0.63) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL678225 0.83 PTGS2 (0.84) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL8442044 0.82 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8483738 0.81 PTGS2 (0.81) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL7175144 0.79 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL8483933 0.79 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL790509 0.78 PTGS2 (0.75) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL15730118 0.78 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL28971530 0.78 MEN1 (0.48) PTGS2PTGS1
SCHEMBL8486254 0.77 PTGS2 (0.74) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106632002-A Preparation technology of etoricoxib and reference substance 5-chloro-3-(4-(methyl sulphonyl)phenyl)-2,3-bipyridine of etoricoxib 贵州大学 2017-05-10 CN disclosed