SCHEMBL28146558

SCHEMBL28146558

COc1ccc2c(c1)CCNC2(C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
RECQL P46063 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
HTR2C P28335 2/20 0.37
HTR2A P28223 1/20 0.37
HTR2B P41595 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
CASP1 P29466 1/20 0.37
BLM P54132 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30931799 0.84 PNMT (0.42) ALDH1A1MAPTRECQLTDP1KDM4E
SCHEMBL17395273 0.83 ALDH1A1 (0.35) ALDH1A1MAPTRECQLTDP1KDM4E
SCHEMBL5211064 0.82 MAPK1 (0.36) ALDH1A1MAPTRECQLTDP1KDM4E
SCHEMBL1202127 0.80 ESR2 (0.41) ALDH1A1MAPTRECQLTDP1KDM4E
SCHEMBL15112425 0.76 MAPKAPK2 (0.47) ALDH1A1MAPTRECQLKDM4ETHRB
SCHEMBL1972155 0.73 MTNR1A (0.39) CASP1MTNR1AMTNR1BSMN1; SMN2ESR1
SCHEMBL715619 0.71 EPHX2 (0.38) ALDH1A1RECQLCYP3A4BLMCYP2C19
SCHEMBL30899459 0.71 EPHX2 (0.38) ALDH1A1RECQLCYP3A4BLMCYP2C19
SCHEMBL304611 0.71 EPHX2 (0.38) ALDH1A1RECQLCYP3A4BLMCYP2C19
SCHEMBL22145508 0.70 KDM1A (0.46) HTR2CHTR2AHTR2BKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106795118-B Heterocyclic compound and their purposes as relevant orphan receptor (ROR) the GAMMA-T inhibitor of retinoids 武田药品工业株式会社 2019-10-08 CN disclosed
CN-106795118-A Heterocyclic compound to they as related orphan receptor (ROR) the GAMMA T inhibitor of retinoids purposes 武田药品工业株式会社 2017-05-31 CN disclosed