SCHEMBL28148240

SCHEMBL28148240

c1cnc(N2CCCC2)c(-c2ccc3ncncc3c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.50
PIK3CD O00329 1/20 0.46
PIK3CA P42336 1/20 0.46
TDO2 P48775 1/20 0.45
METAP2 P50579 3/20 0.41
CYP1A2 P05177 7/20 0.41
CYP3A4 P08684 6/20 0.41
ALDH1A1 P00352 5/20 0.41
TSHR P16473 3/20 0.41
HSD17B10 Q99714 3/20 0.41
CYP2D6 P10635 2/20 0.41
EGFR P00533 2/20 0.39
KDM4E B2RXH2 4/20 0.39
LMNA P02545 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPK1 P28482 3/20 0.39
CLK4 Q9HAZ1 2/20 0.39
ALOX15 P16050 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28148239 0.99 ALOX5AP (0.49) ALOX5APPIK3CDPIK3CATDO2METAP2
SCHEMBL28871485 0.89 CYP2C19 (0.49) PIK3CDPIK3CATDO2METAP2CYP1A2
SCHEMBL28286116 0.89 CYP1A2 (0.55) METAP2CYP1A2CYP3A4ALDH1A1TSHR
SCHEMBL18069431 0.76 PIK3CA (0.52) PIK3CDPIK3CATDO2EGFRKDM4E
SCHEMBL24377491 0.73 ALDH1A1 (0.55) ALOX5APPIK3CACYP1A2CYP3A4ALDH1A1
SCHEMBL27389897 0.72 IP6K1 (0.53) PIK3CDPIK3CAEGFRKDM4E
SCHEMBL28018836 0.72 PIK3CD (0.48) PIK3CDPIK3CATDO2ALDH1A1EGFR
SCHEMBL8870802 0.71 MAP4K4 (0.54) PIK3CDPIK3CAEGFRMAPT
SCHEMBL24196910 0.71 ALOX5AP (0.50) ALOX5APMETAP2CYP1A2CYP3A4ALDH1A1
SCHEMBL28138760 0.71 PIK3CA (0.50) PIK3CDPIK3CATDO2EGFRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106588871-B A kind of 2- substituted pyridinyl quinazolinone analog derivative, its preparation method and use 贵州大学 2019-04-16 CN disclosed
CN-106588871-A 2-substituted pyridyl quinazolinone derivative and synthesis method and application thereof 贵州大学 2017-04-26 CN disclosed