SCHEMBL28151007

SCHEMBL28151007

[N-]=[N+]=NC(=O)c1cccc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.52
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 3/20 0.41
MAPT P10636 2/20 0.41
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
KCNMA1 Q12791 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 1/20 0.40
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28396264 0.87 L3MBTL1 (0.41) PARP1MEN1KMT2AGAAL3MBTL1
SCHEMBL17025091 0.82 PARP1 (0.43) PARP1ERCC5FEN1MEN1KMT2A
SCHEMBL29961790 0.82 PARP1 (0.43) PARP1ERCC5FEN1MEN1KMT2A
SCHEMBL28924563 0.80 PBRM1 (0.52) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL29200432 0.79 CES2 (0.55) PARP1MEN1KMT2ASMN1; SMN2HTT
SCHEMBL29200417 0.79 PARP1 (0.52) PARP1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL19398201 0.79 PARP1 (0.52) PARP1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL13909938 0.77 IDO1 (0.33) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL17454634 0.77 KMO (0.55) ERCC5FEN1MAPTGAA
SCHEMBL30151360 0.77 KMO (0.55) ERCC5FEN1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658868-A Benzamide derivative and preparation method and application thereof 中山大学 2024-03-08 CN disclosed
CN-111662202-B Synthetic method of alpha-ketoamide compound 五邑大学 2022-09-30 CN disclosed
CN-111662202-A Synthetic method of alpha-ketoamide compound 五邑大学 2020-09-15 CN disclosed
CN-106661043-A 2-oxa-5-azabicyclo[2.2.1]heptan-3-yl derivatives 豪夫迈·罗氏有限公司 2017-05-10 CN disclosed