SCHEMBL28152181

SCHEMBL28152181

CC(C)(C)OC(=O)N1CCCC[C@H]1c1nc2ccccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HCRTR1 O43613 2/20 0.46
HCRTR2 O43614 2/20 0.46
PDE10A Q9Y233 1/20 0.46
NPC1 O15118 1/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23247964 1.00 RAB9A (0.47) RAB9ASMN1; SMN2HCRTR1HCRTR2PDE10A
SCHEMBL7329173 0.97 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL7329171 0.97 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL7330933 0.97 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL12509701 0.87 CHEK2 (0.46) HCRTR1HCRTR2
SCHEMBL12327656 0.85 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL12567373 0.85 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL17277682 0.85 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL16215441 0.85 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL15048040 0.84 CHEK2 (0.42) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928126-B Amide derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2019-12-20 CN disclosed
CN-106928126-A A kind of amide derivatives and preparation method thereof and application pharmaceutically 四川海思科制药有限公司 2017-07-07 CN disclosed