SCHEMBL28154690

SCHEMBL28154690

Cc1sc(Nc2cnccn2)nc1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.59
GRM4 Q14833 1/20 0.56
ALDH1A1 P00352 4/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 1/20 0.53
POLB P06746 1/20 0.53
MAOA P21397 11/20 0.52
MAOB P27338 11/20 0.52
MEN1 O00255 2/20 0.52
MAPT P10636 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
GAA P10253 1/20 0.52
CYP2D6 P10635 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ADORA3 P0DMS8 2/20 0.48
ADORA2A P29274 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28155510 0.89 GRM4 (0.50) KDRGRM4ALDH1A1LMNAKDM4E
SCHEMBL367310 0.81 GRM4 (0.72) KDRGRM4ALDH1A1LMNAKDM4E
SCHEMBL369922 0.76 GRM4 (0.67) KDRGRM4ALDH1A1LMNAKDM4E
SCHEMBL12639832 0.74 ALDH1A1 (0.59) ALDH1A1LMNAKDM4EPOLBMAOA
SCHEMBL1745085 0.73 MAOA (0.62) ALDH1A1LMNAMAOAMAOBMEN1
SCHEMBL369152 0.72 GRM4 (1.00) KDRGRM4ALDH1A1LMNAMAOA
SCHEMBL25327043 0.71 MAOA (0.60) ALDH1A1LMNAMAOAMAOBMEN1
SCHEMBL1888443 0.71 NPC1 (0.48) KDRALDH1A1LMNAKDM4EMEN1
SCHEMBL30745793 0.70 GRM4 (0.63) KDRGRM4ALDH1A1LMNAKDM4E
SCHEMBL5174932 0.70 GRM4 (0.63) KDRGRM4ALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254534-B Modulators of HEC1 activity and methods thereof 泰纬生命科技股份有限公司 2017-07-14 CN disclosed