SCHEMBL28158337

SCHEMBL28158337

COc1nc2ccccc2c(Cl)c1Cc1cc2ccccc2s1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.56
CYP2A6 P11509 3/20 0.45
ADRB2 P07550 1/20 0.45
HRH4 Q9H3N8 1/20 0.42
MAPK1 P28482 1/20 0.40
PGK1 P00558 1/20 0.39
ADRA1D P25100 2/20 0.39
AGXT P21549 1/20 0.39
ASIC3 Q9UHC3 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
NR1I3 Q14994 1/20 0.38
PRSS12 P56730 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
KDM1A O60341 1/20 0.36
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36
IDH1 O75874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15648882 0.88 RORC (0.57) RORCCYP2A6ADRB2HRH4PGK1
SCHEMBL16640805 0.80 RORC (0.66) RORC
SCHEMBL16633015 0.76 RORC (0.64) RORC
SCHEMBL16475344 0.75 RORC (0.81) RORC
SCHEMBL16461502 0.71 CYP1A2 (0.45) RORCCYP2A6ADRB2HRH4ADRA1D
SCHEMBL16655564 0.70 RORC (0.59) RORC
SCHEMBL28201461 0.69 CYP2A6 (0.44) RORCCYP2A6ADRB2ADRA1DAGXT
SCHEMBL4961407 0.67 CYP2A6 (0.69) CYP2A6ADRB2ADRA1DAGXTASIC3
SCHEMBL12749518 0.67 CYP1A2 (0.51) RORCMAPK1
SCHEMBL28158505 0.67 CTRC (0.39) RORCCYP2A6ADRB2ADRA1DAGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-B The quinolyl conditioning agent of ROR- γ-T being connect with methylene 詹森药业有限公司 2018-11-09 CN disclosed
CN-105209453-B The quinolyl conditioning agent of the methylene connection of ROR γ T 詹森药业有限公司 2017-06-20 CN disclosed