Bromide

Bromide

SCHEMBL2816388

Br.Br.COc1cc(CNC(=N)S)cc(CNC(=N)S)c1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2A known ✓ Q12879 2/20 0.39
TACR1 P25103 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 4/20 0.40
TSHR P16473 1/20 0.40
PKM P14618 1/20 0.40
HIF1A Q16665 1/20 0.39
GRIN2D O15399 2/20 0.39
GRIN3B O60391 2/20 0.39
GRIN1 Q05586 2/20 0.39
GRIN2B Q13224 2/20 0.39
GRIN2C Q14957 2/20 0.39
GRIN3A Q8TCU5 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MMP13 P45452 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2810051 0.98 TACR1 (0.43) TACR1MEN1KMT2AALDH1A1TSHR
Bromide SCHEMBL28186823 0.83 SMN1; SMN2 (0.58) MEN1KMT2AALDH1A1HTTSMN1; SMN2
SCHEMBL5793985 0.80 ALDH1A1 (0.62) MEN1KMT2AALDH1A1PKMHTT
Bromide SCHEMBL2810233 0.79 PGK1 (0.35) MEN1KMT2AALDH1A1SMN1; SMN2MMP13
Hydrochloric Acid SCHEMBL4801815 0.79 ALDH1A1 (0.61) MEN1KMT2AALDH1A1PKMHTT
Hydrochloric Acid SCHEMBL5398263 0.77 ALDH1A1 (0.59) MEN1KMT2AALDH1A1PKMHTT
SCHEMBL2809139 0.77 PGK1 (0.36) MEN1KMT2AALDH1A1SMN1; SMN2MMP13
Bromide SCHEMBL2811699 0.73 ALDH1A1 (0.50) MEN1KMT2AALDH1A1PKM
Bromide SCHEMBL2809451 0.72 ALDH1A1 (0.49) MEN1KMT2AALDH1A1
SCHEMBL2811627 0.71 ALDH1A1 (0.52) MEN1KMT2AALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100240713-A1 AROMATIC AND HETEROAROMATIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2010-09-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240713-A1 AROMATIC AND HETEROAROMATIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS SLC40A1, PAH, FECH GRIN2A 4573/4885TACR1 870/4885MEN1 933/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.