SCHEMBL28164081

SCHEMBL28164081

NC(=O)c1cccc(CC2CCC(c3ccccc3)CC2)c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.59
OPRD1 P41143 6/20 0.59
OPRK1 P41145 2/20 0.59
KCNH2 Q12809 1/20 0.59
KDM1A O60341 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
MRGPRX4 Q96LA9 1/20 0.48
GAA P10253 1/20 0.48
PARP14 Q460N5 3/20 0.47
PARP1 P09874 2/20 0.47
TNKS O95271 1/20 0.47
CYP2C9 P11712 1/20 0.47
PARP10 Q53GL7 1/20 0.44
DGAT1 O75907 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28164115 0.85 GAA (0.61) KDM1AMAOAGAAPARP14PARP1
SCHEMBL28242711 0.81 OPRM1 (0.59) OPRM1OPRD1OPRK1KCNH2KDM1A
SCHEMBL4974021 0.79 OPRM1 (0.56) OPRM1OPRD1OPRK1KCNH2KDM1A
SCHEMBL22112265 0.79 IDO1 (0.43) CYP2C9
Hydrochloric Acid SCHEMBL6393378 0.78 OPRM1 (0.55) OPRM1OPRD1OPRK1KCNH2KDM1A
SCHEMBL1036815 0.77 PARP1 (0.64) OPRM1OPRD1PARP14PARP1
SCHEMBL27533679 0.77 GBA1 (0.57)
SCHEMBL6429862 0.75 GAA (0.60) OPRM1OPRD1OPRK1KCNH2GAA
SCHEMBL28284087 0.74 PARP14 (0.51) OPRM1OPRD1OPRK1KCNH2KDM1A
SCHEMBL7353600 0.72 EED (0.57) OPRM1OPRD1OPRK1KCNH2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106999450-A immunomodulator 弗莱塞斯生物科学公司 2017-08-01 CN disclosed