SCHEMBL22112265

SCHEMBL22112265

OCc1cccc(C[C@H]2CC[C@H](c3ccccc3)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.43
SLC18A3 Q16572 3/20 0.42
GBA1 P04062 1/20 0.41
DRD2 P14416 2/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
DRD3 P35462 1/20 0.40
ESR1 P03372 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
ESR2 Q92731 1/20 0.40
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL758717 0.87 ENPP2 (0.44) GBA1CHRNB4CHRNA3TSHR
SCHEMBL27533679 0.83 GBA1 (0.57) IDO1SLC18A3GBA1
SCHEMBL17982807 0.80 S1PR1 (0.40) SLC18A3GBA1CHRNB4CHRNA3TSHR
SCHEMBL16957589 0.79 DRD2 (0.55) DRD2CHRNB4CHRNA3DRD3CYP3A4
SCHEMBL16578691 0.79 ESR2 (0.51) SLC18A3DRD2CHRNB4CHRNA3DRD3
SCHEMBL17982840 0.79 S1PR1 (0.42) GBA1DRD2CHRNB4CHRNA3DRD3
SCHEMBL28164081 0.79 OPRM1 (0.59) CYP2C9
SCHEMBL17729950 0.74 ESR2 (0.68) IDO1SLC18A3ESR1CYP3A4CYP2C9
SCHEMBL5756827 0.74 ESR2 (0.68) IDO1SLC18A3ESR1CYP3A4CYP2C9
SCHEMBL10881534 0.74 ESR2 (0.68) IDO1SLC18A3ESR1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020120539-A1 NEW PYRROLIDINE-2-CARBOXYLIC ACID DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-06-18 WO disclosed