SCHEMBL28165447

SCHEMBL28165447

[CH2]C1C=Cc2ccncc2C1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.35
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19979167 0.78 SIGMAR1 (0.39) SIGMAR1CHRNB2CHRNA4
SCHEMBL16892310 0.74 SIGMAR1 (0.32) SIGMAR1CHRNB2CHRNA4
SCHEMBL20661768 0.74 SIGMAR1 (0.32) SIGMAR1CHRNB2CHRNA4
SCHEMBL15479677 0.74 SIGMAR1 (0.32) SIGMAR1CHRNB2CHRNA4
SCHEMBL12286123 0.68 SIGMAR1 (0.33) SIGMAR1CHRNB2CHRNA4
SCHEMBL14725544 0.68 CYP11B2 (0.38) SIGMAR1CHRNB2CHRNA4
SCHEMBL4624876 0.66
SCHEMBL16258601 0.63 SIGMAR1 (0.39) SIGMAR1CHRNB2CHRNA4
SCHEMBL30825565 0.63 SIGMAR1 (0.35) SIGMAR1CHRNB2CHRNA4
SCHEMBL1950016 0.63 SIGMAR1 (0.43) SIGMAR1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103958478-B Bicyclic dihydroisoquinolin-1-one derivatives 霍夫曼-拉罗奇有限公司 2017-08-01 CN disclosed