SCHEMBL28165692

SCHEMBL28165692

O=CC(F)(F)F.c1cc2cc-2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.39
PTPN5 P54829 5/20 0.39
MEN1 O00255 1/20 0.39
ESR1 P03372 1/20 0.39
KMT2A Q03164 1/20 0.39
DHODH Q02127 1/20 0.38
KIF11 P52732 2/20 0.37
APP P05067 1/20 0.37
KMO O15229 1/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
DRD1 P21728 1/20 0.35
AGXT P21549 1/20 0.35
ERN1 O75460 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL26134410 0.81 KIF11 (0.56) PTPN1PTPN5KIF11CYP1A2CYP3A4
SCHEMBL27798276 0.77 MEN1 (0.46) PTPN1MEN1ESR1KMT2AAPP
SCHEMBL308018 0.77 NFE2L2 (0.46) PTPN1CYP1A2CYP3A4CYP2D6
SCHEMBL7946647 0.75 ESR1 (0.41) MEN1ESR1KMT2ADHODHKIF11
Formic Acid SCHEMBL3169782 0.75
Acetaldehyde SCHEMBL895439 0.75
SCHEMBL28211296 0.74 DRD1 (0.43) MEN1ESR1KMT2AAPPKMO
Benzene SCHEMBL21296191 0.73 KIF11 (0.30) KIF11CYP2A6
SCHEMBL7196829 0.73
SCHEMBL4969576 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107011138-A A kind of preparation method of sitagliptin intermediate 江苏汉阔生物有限公司 2017-08-04 CN claimed
CN-107501112-B A kind of Chiral Synthesis of chiral beta-amino acids and the synthetic method of medicine intermediate 苏州爱玛特生物科技有限公司 2019-06-11 CN disclosed
CN-105330664-B A kind of synthetic method of Xi Gelieting impurity 合肥华方医药科技有限公司 2018-06-19 CN disclosed
CN-107501112-A A kind of Chiral Synthesis of chiral beta amino acids and the synthetic method of medicine intermediate 苏州爱玛特生物科技有限公司 2017-12-22 CN disclosed
CN-107011138-A A kind of preparation method of sitagliptin intermediate 江苏汉阔生物有限公司 2017-08-04 CN disclosed