Indole

Indole

SCHEMBL28167409

NC(=O)N1CC=Cc2ccccc21.c1ccc2[nH]ccc2c1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ITGB2 P05107 1/20 0.44
ICAM1 P05362 1/20 0.44
ITGAL P20701 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
AHR P35869 1/20 0.44
ADK P55263 1/20 0.44
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
SCN4A P35499 1/20 0.41
SCN5A Q14524 1/20 0.41
SCN9A Q15858 1/20 0.41
P2RX4 Q99571 5/20 0.38
PDPK1 O15530 1/20 0.33
AMPD2 Q01433 3/20 0.32
FGFR1 P11362 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indole SCHEMBL28214491 0.88 TRPA1 (0.45) TRPA1CA1CA2ITGB2ICAM1
SCHEMBL1286806 0.85 LMNA (0.55) LMNATSHRMAPK1SCN4ASCN5A
Hydrochloric Acid SCHEMBL28145471 0.83 LMNA (0.53) LMNATSHRMAPK1SCN4ASCN5A
Indole SCHEMBL27827279 0.81 TRPA1 (0.38) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL28196583 0.80 TRPA1 (0.50) TRPA1CA1CA2ITGB2ICAM1
SCHEMBL28205987 0.78 P2RX4 (0.40) LMNATSHRMAPK1SCN4ASCN5A
SCHEMBL28081008 0.77 KDM4E (0.38) LMNATSHRMAPK1SCN4ASCN5A
Isoquinoline SCHEMBL28191779 0.76 LMNA (0.40) LMNATSHRMAPK1SCN4ASCN5A
Indole SCHEMBL5205084 0.73 TRPA1 (0.74) TRPA1CA1CA2ITGB2ICAM1
Indole SCHEMBL27631042 0.73 TRPA1 (0.74) TRPA1CA1CA2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073741-B Phthalazinones and isoquinolinones as ROCK inhibitors 百时美施贵宝公司 2017-08-08 CN disclosed