SCHEMBL2817256

SCHEMBL2817256

CN(C)C(C(N)=O)c1cccc2[nH]cnc12

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.54
ALDH1A1 P00352 2/20 0.37
PKM P14618 1/20 0.37
LMNA P02545 2/20 0.35
TSHR P16473 2/20 0.35
PAX8 Q06710 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MMP9 P14780 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BRD4 O60885 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2820806 0.82 PARP1 (0.56) PARP1BRD4
SCHEMBL7032508 0.79 PARP1 (0.52) PARP1
SCHEMBL2817264 0.79 PARP1 (0.34) PARP1ALDH1A1LMNATSHRPAX8
SCHEMBL2497545 0.75 PARP1 (0.50) PARP1BRD4
SCHEMBL7856459 0.73 PARP1 (0.47) PARP1ALDH1A1PKMLMNAKDM4E
SCHEMBL2611049 0.73 PARP1 (0.46) PARP1ALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL2128641 0.72 ALDH1A1 (0.40) PARP1ALDH1A1PKMBRD4
SCHEMBL24351926 0.70 PARP1 (0.44) PARP1ALDH1A1LMNASMN1; SMN2BRD4
SCHEMBL630485 0.70 PARP1 (1.00) PARP1
SCHEMBL2127994 0.70 HTR2A (0.47) PARP1LMNABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010110686-A1 PYRIMIDINYL AND 1,3,5 TRIAZINYL BENZIMIDAZOLES AND THEIR USE IN CANCER THERAPY PATHWAY THERAPEUTICS LIMITED (NZ) 2010-09-30 WO disclosed