SCHEMBL28182115

SCHEMBL28182115

COc1ccc(-c2ncsc2-c2ccc3nccnc3c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
KMT2A Q03164 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
STAT1 P42224 1/20 0.43
CCNB2 O95067 1/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL926052 0.83 ALDH1A1 (0.50) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL28182976 0.81 FLT3 (0.44) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL28950139 0.78 DYRK1A (0.61) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL18041689 0.78 TGFBR1 (0.61) MAPTNPC1RAB9AKDM4EALDH1A1
Alcohol SCHEMBL11561027 0.77 ALDH1A1 (0.44) MAPTKDM4EALDH1A1KMT2AMEN1
SCHEMBL28182986 0.74 TGFBR1 (0.47) MAPTKDM4EKMT2AMEN1TGFBR1
SCHEMBL28182113 0.71 TGFBR1 (0.51) TGFBR1MAPK14
SCHEMBL622115 0.71 KDM4E (0.56) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL29550130 0.71 KDM4E (0.56) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL4035268 0.69 TGFBR1 (0.60) TGFBR1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107406412-A TGF beta inhibitors 里格尔药品股份有限公司 2017-11-28 CN claimed
CN-107406412-A TGF beta inhibitors 里格尔药品股份有限公司 2017-11-28 CN disclosed