SCHEMBL926052

SCHEMBL926052

COc1ccc(-c2ncsc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
KDM4E B2RXH2 5/20 0.50
MAPT P10636 4/20 0.50
KMT2A Q03164 2/20 0.46
PTGS2 P35354 2/20 0.46
HPGD P15428 2/20 0.45
LMNA P02545 3/20 0.44
GAA P10253 2/20 0.44
CLK4 Q9HAZ1 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
ADORA1 P30542 1/20 0.42
APP P05067 1/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alcohol SCHEMBL11561027 0.92 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTKMT2APTGS2
SCHEMBL28182115 0.83 MAPT (0.43) ALDH1A1KDM4EMAPTKMT2AHPGD
SCHEMBL16300950 0.81 ALOX5 (0.49) ALDH1A1KDM4EMAPTKMT2APTGS2
SCHEMBL31609684 0.80 KMT2A (0.45) ALDH1A1KDM4EMAPTKMT2APTGS2
SCHEMBL9256402 0.80 KMT2A (0.45) ALDH1A1KDM4EMAPTKMT2APTGS2
SCHEMBL2088457 0.77 PTGS2 (0.42) ALDH1A1KDM4EMAPTKMT2APTGS2
SCHEMBL5815370 0.76 POLB (0.40) ALDH1A1KDM4EMAPTKMT2AHPGD
SCHEMBL2088458 0.76 PTGS2 (0.41) ALDH1A1KDM4EMAPTPTGS2LMNA
SCHEMBL5813457 0.74 NPC1 (0.39) ALDH1A1KDM4EMAPTKMT2AHPGD
SCHEMBL926914 0.74 KDM4E (0.55) ALDH1A1KDM4EMAPTGAAADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 103 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4168315-A ANTICOAGULANTS THE UPJOHN COMPANY (US) 1979-09-18 US claimed
EP-2006738-B1 Lithographic printing plate precursor FUJIFILM CORP (JP) 2017-09-06 EP disclosed
EP-2259141-B1 PROCESS FOR PRODUCING LITHOGRAPHIC PRINTING PLATE FUJIFILM CORP (JP) 2016-11-23 EP disclosed
EP-1939687-B1 Polymerizable composition and lithographic printing plate precursor FUJIFILM CORP (JP) 2016-09-14 EP disclosed
EP-2503393-B2 Method for preparation of lithographic printing plate FUJIFILM CORP (JP) 2016-07-20 EP disclosed
EP-2042312-B1 Processing method of lithographic printing plate precursor FUJIFILM CORP (JP) 2016-05-18 EP disclosed
EP-3021167-A1 LITHOGRAPHIC PRINTING PLATE PRECURSOR AND METHOD OF PREPARING LITHOGRAPHIC PRINTING PLATE Fujifilm Corporation (JP) 2016-05-18 EP disclosed
EP-2045662-B1 Lithographic printing plate precursor and method of preparing lithographic printing plate FUJIFILM CORP (JP) 2015-12-23 EP disclosed
EP-1975708-B1 Lithographic printing plate precursor FUJIFILM CORP (JP) 2015-04-22 EP disclosed
EP-2662729-B1 Method for preparation of lithographic printing plate FUJIFILM CORP (JP) 2014-10-22 EP disclosed
EP-0772606-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
WO-1996003392-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed
EP-0159677-B1 NOVEL 4,5-BIS(4-METHOXYPHENYL)-2-(PYRROL-2-YL)THIAZOLES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME KANEBO, LTD. (JP) 1989-02-22 EP disclosed
US-4659726-A ANTICOAGULANTS KANEBO, LTD. (JP) 1987-04-21 US disclosed
EP-0159677-A2 Novel 4,5-bis(4-methoxyphenyl)-2-(pyrrol-2-yl)thiazoles, process for the preparation thereof and pharmaceutical composition containing the same KANEBO, LTD. (JP) 1985-10-30 EP disclosed
US-4451471-A Certain 2,4,5-tri-substituted thiazoles, pharmaceutical compositions containing same and methods of using same CIBA-GEIGY CORPORATION (US) 1984-05-29 US disclosed
EP-0061425-A2 Thiazole derivatives, processes for their preparation, medicaments containing them and their use CIBA-GEIGY AG (CH) 1982-09-29 EP disclosed
US-4322428-A 2(4-Fluorophenyl)-4,5,-bis(4-methoxyphenyl)thiazole and method of use ELI LILLY AND COMPANY (US) 1982-03-30 US disclosed
EP-0037274-A1 Substituted triaryl thiazole compounds ELI LILLY AND COMPANY (US) 1981-10-07 EP disclosed
US-4168315-A ANTICOAGULANTS THE UPJOHN COMPANY (US) 1979-09-18 US disclosed