SCHEMBL28189028

SCHEMBL28189028

O=C(O)C12CC3CC(C1)C(c1ccc(O)cc1)C(C3)C2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.57
CYP2C9 P11712 1/20 0.57
ESR2 Q92731 1/20 0.57
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
XBP1 P17861 1/20 0.46
HSD11B1 P28845 5/20 0.41
HSD11B2 P80365 4/20 0.41
HSP90AA1 P07900 1/20 0.41
P2RX7 Q99572 2/20 0.40
CNR2 P34972 1/20 0.39
DGAT1 O75907 4/20 0.38
EPHX2 P34913 1/20 0.37
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18007733 0.87 HSD11B1 (0.49) ESR1CYP2C9ESR2HSD11B1HSD11B2
SCHEMBL27713466 0.78 MAPK1 (0.43) ESR1CYP2C9ESR2MAPTHSD11B1
SCHEMBL31042568 0.77 ESR2 (0.64) ESR1CYP2C9ESR2GAAMAPT
SCHEMBL3644747 0.75 HSD11B1 (0.43) HSD11B1HSD11B2DGAT1KDM4EALDH1A1
SCHEMBL19798638 0.75 MAPK1 (0.42) ESR1CYP2C9ESR2MAPTHSD11B1
SCHEMBL16902818 0.74 ESR1 (0.60) ESR1CYP2C9ESR2GAAMAPT
SCHEMBL30215621 0.73 ESR2 (1.00) ESR1CYP2C9ESR2GAAMAPT
SCHEMBL22191212 0.73 HSP90AA1 (0.52) ESR1ESR2GAAMAPTXBP1
SCHEMBL3148759 0.72 ESR2 (0.56) ESR1CYP2C9ESR2GAAMAPT
SCHEMBL3192560 0.71 HSD11B1 (0.60) HSD11B1HSD11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107438611-B fused ring compound, pharmaceutical composition and application thereof SHANGHAI DE NOVO PHARMATECH CO.,LTD. (CN) 2019-10-29 CN disclosed
CN-107438611-A fused ring compound, pharmaceutical composition and application thereof 上海迪诺医药科技有限公司 2017-12-05 CN disclosed