SCHEMBL28192142

SCHEMBL28192142

C1=c2ccccc2=NC(c2cccnc2)N1c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
HTT P42858 2/20 0.44
MAPK1 P28482 1/20 0.44
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
NPEPPS P55786 1/20 0.37
TP53 P04637 1/20 0.36
MDM2 Q00987 1/20 0.36
NPSR1 Q6W5P4 2/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP11B2 P19099 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10957215 0.87 ALDH1A1 (0.32) ALDH1A1GAA
SCHEMBL28192758 0.85 MAPT (0.43) MAPTHTTMAPK1ALDH1A1GAA
SCHEMBL28192154 0.84 MAPT (0.41) MAPTALDH1A1TP53NPSR1
SCHEMBL30913234 0.82 L3MBTL1 (0.34) MAPTHTTMAPK1ALDH1A1CYP2A6
SCHEMBL28324686 0.77 ALDH1A1 (0.38) MAPTHTTALDH1A1GAANPSR1
SCHEMBL28324633 0.77 GAA (0.35) MAPTMAPK1ALDH1A1GAATDP1
SCHEMBL28324627 0.77 GAA (0.38) MAPTMAPK1ALDH1A1GAATDP1
SCHEMBL28192176 0.77 PRKCZ (0.38) MAPTGAA
SCHEMBL28192157 0.77 KMT2A (0.38) MAPTMAPK1ALDH1A1GAA
SCHEMBL28854127 0.76 L3MBTL1 (0.39) MAPTHTTALDH1A1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN claimed
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN disclosed