SCHEMBL28192561

SCHEMBL28192561

COC(=O)C(CN)c1cccc(F)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.48
AOC3 Q16853 1/20 0.48
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
KDM4E B2RXH2 1/20 0.45
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
CNR2 P34972 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KCNQ2 O43526 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17825651 0.87 ROCK2 (0.45) ROCK2AOC3HDAC4HDAC7HDAC5
SCHEMBL31038318 0.86 HDAC4 (0.47) ROCK2AOC3HDAC4HDAC7HDAC5
SCHEMBL25242939 0.86 HDAC4 (0.47) ROCK2AOC3HDAC4HDAC7HDAC5
Hydrochloric Acid SCHEMBL7339178 0.85 ROCK2 (0.44) ROCK2AOC3HDAC4HDAC7HDAC5
Hydrochloric Acid SCHEMBL7379790 0.85 ROCK2 (0.44) ROCK2AOC3HDAC4HDAC7HDAC5
Hydrochloric Acid SCHEMBL7379773 0.85 ROCK2 (0.44) ROCK2AOC3HDAC4HDAC7HDAC5
SCHEMBL12073600 0.85 HDAC4 (0.46) AOC3HDAC4HDAC7HDAC5KDM4E
SCHEMBL20826236 0.82 HDAC4 (0.44) AOC3HDAC4HDAC7HDAC5KDM4E
SCHEMBL17798382 0.82 ALDH1A1 (0.42) ROCK2KDM4EKMT2A
SCHEMBL30932899 0.82 L3MBTL1 (0.55) ROCK2AOC3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107522634-A Biaryl ureas carboxylic acid derivates or its salt and its production and use 复旦大学 2017-12-29 CN disclosed