SCHEMBL28199441

SCHEMBL28199441

Cc1c(N=O)ccc2[nH]ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
P2RX7 Q99572 2/20 0.36
AHR P35869 1/20 0.34
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31
GLA P06280 2/20 0.31
CYP3A4 P08684 2/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
DYRK1A Q13627 1/20 0.31
HASPIN Q8TF76 1/20 0.31
DYRK2 Q92630 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404367 0.73 AHR (0.40) PARP1P2RX7AHRHTR1DHTR1B
SCHEMBL4572244 0.72 AHR (0.50) AHRRHEB
SCHEMBL13820047 0.71 P2RX7 (0.40) PARP1P2RX7AHRMTNR1AMTNR1B
SCHEMBL16366637 0.70 MTNR1A (0.36) P2RX7KDM4EGLAHSD17B10KMT2A
SCHEMBL724626 0.69 AHR (0.38) PARP1P2RX7AHRALDH1A1KDM4E
SCHEMBL8995172 0.69 AHR (0.52) PARP1P2RX7AHRHTR1DHTR1B
SCHEMBL28142795 0.69 AHR (0.38) PARP1P2RX7AHRMTNR1AMTNR1B
SCHEMBL2976758 0.69 AHR (0.38) PARP1P2RX7AHRHTR1DHTR1B
SCHEMBL31005469 0.69 P2RX7 (0.38) PARP1P2RX7AHRALDH1A1KDM4E
SCHEMBL2120711 0.69 PARP1 (0.40) PARP1P2RX7AHRDYRK1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492434-B Miscellaneous bicyclic aryl RORC2 inhibitor and its application method 辉瑞大药厂 2018-02-16 CN disclosed