SCHEMBL28200313

SCHEMBL28200313

O=c1cc(-c2cccc(C(F)(F)F)c2)nc[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.59
KMO O15229 2/20 0.52
IDO1 P14902 1/20 0.51
CTSS P25774 3/20 0.49
CTSK P43235 2/20 0.49
MAOB P27338 1/20 0.48
NOTUM Q6P988 1/20 0.48
SCN2A Q99250 2/20 0.47
MAPT P10636 1/20 0.46
KDR P35968 1/20 0.46
MAPK14 Q16539 1/20 0.46
TNNI3K Q59H18 1/20 0.46
PIM1 P11309 2/20 0.45
PARP1 P09874 1/20 0.44
MAP4K4 O95819 1/20 0.44
GPX4 P36969 1/20 0.44
GSK3B P49841 1/20 0.44
PIM3 Q86V86 1/20 0.44
BRSK1 Q8TDC3 1/20 0.44
MAP4K5 Q9Y4K4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4058328 0.84 PDE2A (0.47) XDHMAOBNOTUMPARP1GSK3B
SCHEMBL3451431 0.78 XDH (0.49) XDHKMONOTUMMAPTGSK3B
SCHEMBL28199707 0.78 XDH (0.62) XDHCTSSCTSK
SCHEMBL311778 0.78 IDO1 (0.54) XDHKMOIDO1CTSSCTSK
Hydrochloric Acid SCHEMBL29856925 0.76 XDH (0.47) XDHKMONOTUMMAPTGSK3B
SCHEMBL29417235 0.75 TRPV4 (0.44) MAP4K4
SCHEMBL1769732 0.75 JAK2 (0.62) XDHKMOIDO1CTSSMAOB
SCHEMBL7782564 0.74 DAO (0.49) KDRMAPK14TNNI3K
SCHEMBL11515630 0.73 IDO1 (0.60) XDHKMOIDO1CTSSMAOB
SCHEMBL6284522 0.71 DGAT1 (0.52) XDHIDO1MAOBNOTUMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860937-B Suppress the compound of function with beta-secretase, prepare method of the compound and application thereof 北京大学 2018-02-06 CN disclosed