SCHEMBL28200773

SCHEMBL28200773

CS(=O)(=O)c1ccc(C[CH]N2CCOCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.49
ALDH1A1 P00352 1/20 0.43
TSHR P16473 2/20 0.42
PKM P14618 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 3/20 0.40
GHSR Q92847 1/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 1/20 0.39
KCNJ1 P48048 1/20 0.39
KCNH2 Q12809 1/20 0.39
PIK3CA P42336 2/20 0.39
PIK3CG P48736 2/20 0.39
RORC P51449 1/20 0.38
POLB P06746 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL946953 0.77 LMNA (0.50) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL5776873 0.76 HRH3 (0.61) AKR1C3ALDH1A1TSHRMEN1KMT2A
SCHEMBL5776872 0.76 AKR1C3 (0.49) AKR1C3ALDH1A1TSHRPKMMEN1
SCHEMBL6867994 0.75 AKR1C3 (0.71) AKR1C3ALDH1A1TSHRPKMMEN1
SCHEMBL28205415 0.72 ALDH1A1 (0.45) AKR1C3ALDH1A1PKMMEN1KMT2A
SCHEMBL28140146 0.72 ALDH1A1 (0.56) AKR1C3ALDH1A1TSHRMEN1KMT2A
SCHEMBL31482340 0.71 ALDH1A1 (0.51) AKR1C3ALDH1A1TSHRMEN1KMT2A
SCHEMBL4397821 0.71 ALDH1A1 (0.67) AKR1C3ALDH1A1MEN1KMT2AGAA
SCHEMBL1428902 0.70 ENPP2 (0.48) AKR1C3KCNJ1KCNH2
SCHEMBL12793723 0.70 POLB (0.73) ALDH1A1TSHRMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107641089-A A kind of preparation method of the mesyl phenylacetic acid of Etoricoxib intermediate 4 天津药物研究院有限公司 2018-01-30 CN claimed
CN-107641089-A A kind of preparation method of the mesyl phenylacetic acid of Etoricoxib intermediate 4 天津药物研究院有限公司 2018-01-30 CN disclosed