SCHEMBL28203407

SCHEMBL28203407

O=c1cc(-c2cc(Cl)ccc2C(F)F)cc[nH]1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.44
HDAC6 Q9UBN7 2/20 0.43
NOTUM Q6P988 1/20 0.41
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PPOX P50336 1/20 0.39
S100A4 P26447 2/20 0.38
AOC3 Q16853 2/20 0.37
F11 P03951 1/20 0.37
ALDH2 P05091 5/20 0.36
KCNH2 Q12809 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SCN8A Q9UQD0 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475271 0.77 AHR (0.50) MAP4K4NOTUMPDE3BPDE3APPOX
SCHEMBL16115826 0.76 F11 (0.39) MAP4K4PDE3BPDE3APPOXS100A4
SCHEMBL31252350 0.73 F11 (0.42) HDAC6AOC3F11
SCHEMBL3476831 0.71 NOTUM (0.64) MAP4K4NOTUMAOC3ALDH2KCNH2
SCHEMBL3477513 0.71 MAP4K4 (0.45) MAP4K4NOTUMPDE3BPDE3ASCN8A
SCHEMBL16115727 0.71 F11 (0.44) S100A4F11
SCHEMBL17629754 0.71 NR3C1 (0.38) S100A4F11ALDH1A1SCN8ASCN10A
SCHEMBL16144671 0.69 F11 (0.45) MAP4K4F11
SCHEMBL19620153 0.69 MAP4K4 (0.43) MAP4K4NOTUMPDE3BPDE3APPOX
SCHEMBL608199 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108164513-A Substituted oxo pyridine derivative and its purposes in terms of cardiovascular disorder is treated 拜耳制药股份公司 2018-06-15 CN disclosed
CN-105164122-B Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders 拜耳制药股份公司 2018-02-02 CN disclosed