SCHEMBL28204604

SCHEMBL28204604

CCCCc1c(F)cccc1C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 7/20 0.45
CYP3A4 P08684 3/20 0.44
MEN1 O00255 1/20 0.44
NR1I2 O75469 1/20 0.44
LMNA P02545 1/20 0.44
CHRM2 P08172 1/20 0.44
ADRA2A P08913 1/20 0.44
MAPT P10636 1/20 0.44
OPRK1 P41145 1/20 0.44
HTR2B P41595 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
MAPK8 P45983 2/20 0.43
MC4R P32245 1/20 0.41
KCNH2 Q12809 1/20 0.40
PLK1 P53350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21439307 0.90 MAPK8 (0.44) CD38CYP3A4MEN1NR1I2LMNA
SCHEMBL2972655 0.88 LMNA (0.50) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL27556126 0.83 CYP3A4 (0.46) CD38CYP3A4MEN1NR1I2LMNA
SCHEMBL30499962 0.83 MAPK8 (0.47) CD38CYP3A4MEN1NR1I2LMNA
SCHEMBL19695740 0.83 MAPK8 (0.47) CD38CYP3A4MEN1NR1I2LMNA
SCHEMBL5370893 0.83 CYP3A4 (0.53) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL6258469 0.82 ALDH1A1 (0.46) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL6285466 0.82 CYP3A4 (0.45) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL28293673 0.82 MEN1 (0.41) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL6535320 0.81 LMNA (0.55) CYP3A4MEN1NR1I2LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104341351-B A kind of Diarylthiohydantoin derivative and its application 北京海美源医药科技有限公司 2018-02-06 CN disclosed