SCHEMBL28205358

SCHEMBL28205358

NC(=O)c1ccc2c(c1)CN(C(=O)O)C2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.49
HSD17B3 P37058 1/20 0.48
HDAC6 Q9UBN7 4/20 0.45
HDAC8 Q9BY41 3/20 0.45
KDM1A O60341 2/20 0.42
ENPP2 Q13822 1/20 0.40
DPP9 Q86TI2 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TSHR P16473 1/20 0.40
OPRM1 P35372 1/20 0.38
PLAU P00749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075113 0.85 ALDH1A1 (0.53) NAMPTHDAC6HDAC8ALDH1A1KDM4E
SCHEMBL14590639 0.84 HSD17B3 (0.57) NAMPTHSD17B3HDAC6HDAC8KDM1A
SCHEMBL26075696 0.80 HSD17B3 (0.52) NAMPTHSD17B3HDAC6HDAC8KDM1A
SCHEMBL28956614 0.79 HDAC6 (0.50) NAMPTHDAC6HDAC8
SCHEMBL29168673 0.78 HDAC6 (0.56) NAMPTHDAC6HDAC8DPP9ALDH1A1
SCHEMBL1027717 0.78 NAMPT (0.54) NAMPTHDAC6HDAC8ALDH1A1KDM4E
SCHEMBL1393814 0.78 NR1H2 (0.50) NAMPTHSD17B3HDAC6HDAC8DPP9
SCHEMBL14625863 0.77 HSD17B3 (0.50) NAMPTHSD17B3HDAC6HDAC8KDM1A
SCHEMBL566491 0.77 HDAC6 (0.51) NAMPTHDAC6HDAC8
SCHEMBL4232286 0.77 NR1H2 (0.56) NAMPTHSD17B3HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849047-A Biphenyl derivative, preparation method and medical application thereof 四川海思科制药有限公司 2018-03-27 CN disclosed