SCHEMBL1075113

SCHEMBL1075113

O=C(O)c1ccc2c(c1)CN(C(=O)O)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
NAMPT P43490 3/20 0.49
HDAC6 Q9UBN7 4/20 0.47
HDAC8 Q9BY41 2/20 0.47
SRD5A2 P31213 4/20 0.47
MYC P01106 1/20 0.45
SRD5A1 P18405 3/20 0.43
KDM4E B2RXH2 4/20 0.42
MAPT P10636 4/20 0.42
POLB P06746 2/20 0.42
BLM P54132 1/20 0.42
GRM1 Q13255 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28052395 0.86 MYC (0.56) ALDH1A1HDAC6HDAC8MYCMEN1
SCHEMBL28205358 0.85 NAMPT (0.49) ALDH1A1NAMPTHDAC6HDAC8KDM4E
SCHEMBL7277193 0.85 NOTUM (0.58) ALDH1A1NAMPTHDAC6HDAC8SRD5A2
SCHEMBL28956614 0.82 HDAC6 (0.50) NAMPTHDAC6HDAC8
SCHEMBL29168673 0.81 HDAC6 (0.56) ALDH1A1NAMPTHDAC6HDAC8
SCHEMBL1027717 0.81 NAMPT (0.54) ALDH1A1NAMPTHDAC6HDAC8KDM4E
SCHEMBL19339147 0.81 ALDH1A1 (0.53) ALDH1A1NAMPTHDAC6HDAC8SRD5A2
SCHEMBL3313453 0.81 ALDH1A1 (0.53) ALDH1A1NAMPTHDAC6HDAC8SRD5A2
SCHEMBL566491 0.80 HDAC6 (0.51) NAMPTHDAC6HDAC8
SCHEMBL2814463 0.79 KMT2A (0.57) ALDH1A1MAPTPOLBMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023284651-A1 N-(2-AMINOPHENYL)BENZAMIDE COMPOUND AND APPLICATION THEREOF 南京明德新药研发有限公司 2023-01-19 WO disclosed
CN-1889970-B Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of HCV replication INTERMUNE INC 2012-06-13 CN disclosed
EP-2274283-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2011-01-19 EP disclosed
WO-2009112550-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2009-09-17 WO disclosed
CN-1889970-A Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of HCV replication INTERMUNE INC (US) 2007-01-03 CN disclosed