SCHEMBL28205403

SCHEMBL28205403

COC(=O)C(Cc1ccc(CCO)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.56
CTSS P25774 8/20 0.51
CTSK P43235 7/20 0.51
CTSB P07858 2/20 0.50
CTSL P07711 1/20 0.50
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
ACE P12821 1/20 0.48
ITGA4 P13612 2/20 0.46
ITGB7 P26010 2/20 0.46
ALDH1A1 P00352 1/20 0.46
THRB P10828 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
EPHX2 P34913 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
AKT1 P31749 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20415892 1.00 KLK5 (0.56) KLK5CTSSCTSKCTSBCTSL
SCHEMBL8234790 0.89 KLK5 (0.61) KLK5CTSSCTSKCTSBCTSL
SCHEMBL4925498 0.89 KLK5 (0.61) KLK5CTSSCTSKCTSBCTSL
SCHEMBL7896684 0.88 KLK5 (0.67) KLK5CTSSCTSKCTSBCTSL
SCHEMBL7544681 0.88 KLK5 (0.57) KLK5CTSSCTSKCTSBCTSL
SCHEMBL18262437 0.88 ACE (0.61) CTSSCTSKCTSBCTSLITGB3
SCHEMBL18262439 0.88 ACE (0.61) CTSSCTSKCTSBCTSLITGB3
SCHEMBL7541415 0.87 KLK5 (0.54) KLK5CTSSCTSKCTSBCTSL
SCHEMBL12035376 0.86 KLK5 (0.58) KLK5CTSSCTSKCTSBCTSL
SCHEMBL539575 0.86 CTSS (0.66) KLK5CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107848962-B Urea derivative or pharmacologically acceptable salt thereof 杏林制药株式会社 2021-04-09 CN disclosed
CN-107848962-A UREA DERIVATIVE OR PHARMACOLOGICALLY ACCEPTABLE SALT THEREOF 杏林制药株式会社 2018-03-27 CN disclosed