SCHEMBL7541415

SCHEMBL7541415

COC(=O)CCc1ccc(CC(NC(=O)OC(C)(C)C)C(=O)OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.54
CTSS P25774 8/20 0.49
CTSK P43235 7/20 0.49
ACE P12821 1/20 0.49
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
ITGA4 P13612 1/20 0.45
ITGB7 P26010 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
EPHX2 P34913 1/20 0.43
ABCB1 P08183 1/20 0.43
HDAC8 Q9BY41 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7544681 0.91 KLK5 (0.57) KLK5CTSSCTSKACECTSL
SCHEMBL20415892 0.87 KLK5 (0.56) KLK5CTSSCTSKACECTSL
SCHEMBL28205403 0.87 KLK5 (0.56) KLK5CTSSCTSKACECTSL
SCHEMBL14021754 0.87 ACE (0.57) CTSSCTSKACECTSLCTSB
SCHEMBL4608263 0.87 ACE (0.57) CTSSCTSKACECTSLCTSB
SCHEMBL7896684 0.86 KLK5 (0.67) KLK5CTSSCTSKACECTSL
SCHEMBL4929625 0.85 KLK5 (0.52) KLK5CTSSCTSKACECTSL
SCHEMBL8232304 0.85 KLK5 (0.52) KLK5CTSSCTSKACECTSL
SCHEMBL4608329 0.85 ITGB3 (0.58) CTSSCTSKACECTSLCTSB
SCHEMBL14021672 0.85 ITGB3 (0.58) CTSSCTSKACECTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1376143-A Carboxylic acid derivatives and adhesion molecule inhibitors containing the same as the active ingredient TORAY INDUSTRIES (JP) 2002-10-23 CN disclosed
EP-1209147-A1 CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2002-05-29 EP disclosed