SCHEMBL28208293

SCHEMBL28208293

C[C@H](N)c1ccc(CN2CCNCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
CXCR4 P61073 12/20 0.56
HRH3 Q9Y5N1 2/20 0.56
MEN1 O00255 1/20 0.56
CHRM2 P08172 1/20 0.56
CHRM1 P11229 1/20 0.56
ADRA2C P18825 1/20 0.56
CCR2 P41597 1/20 0.56
CXCL12 P48061 1/20 0.56
BLM P54132 1/20 0.56
KMT2A Q03164 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
HTR6 P50406 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28208297 1.00 SIGMAR1 (0.56) SIGMAR1CXCR4HRH3MEN1CHRM2
SCHEMBL12015808 0.86 SIGMAR1 (0.59) SIGMAR1CXCR4HRH3MEN1CHRM2
Tert-Butyl Formate SCHEMBL28277618 0.85 CXCR4 (0.43) SIGMAR1CXCR4HRH3MEN1CHRM2
Tert-Butyl Formate SCHEMBL28277617 0.85 CXCR4 (0.43) SIGMAR1CXCR4HRH3MEN1CHRM2
Hydrochloric Acid SCHEMBL29206910 0.85 CXCR4 (0.60) SIGMAR1CXCR4HRH3MEN1CHRM2
SCHEMBL1935806 0.84 HRH3 (0.67) HRH3MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL14847024 0.84 HRH3 (0.67) HRH3MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL12017823 0.82 SIGMAR1 (0.54) SIGMAR1CXCR4HRH3MEN1CHRM2
SCHEMBL24307315 0.81 ALDH1A1 (0.61) HRH3MEN1KMT2AHTR6ALDH1A1
SCHEMBL21378560 0.81 LMNA (0.64) SIGMAR1HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849059-A 7-phenylethylamino-4H-pyrimido [4,5-D ] [1,3] oxazin-2-one compounds and their use as inhibitors of mutant IDH1 伊莱利利公司 2018-03-27 CN disclosed