SCHEMBL2820937

SCHEMBL2820937

CN(C)C(=O)c1cc(Br)cc(C(=O)NC2CC2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 2/20 0.55
TUBB P07437 2/20 0.55
TUBA3C P0DPH7 2/20 0.55
TUBA1B P68363 2/20 0.55
TUBA4A P68366 2/20 0.55
TUBB4B P68371 2/20 0.55
TUBB3 Q13509 2/20 0.55
TUBB2A Q13885 2/20 0.55
TUBB8 Q3ZCM7 2/20 0.55
TUBA3E Q6PEY2 2/20 0.55
TUBA1A Q71U36 2/20 0.55
TUBA1C Q9BQE3 2/20 0.55
TUBB6 Q9BUF5 2/20 0.55
TUBB2B Q9BVA1 2/20 0.55
TUBB1 Q9H4B7 2/20 0.55
SMYD3 Q9H7B4 4/20 0.48
NCEH1 Q6PIU2 3/20 0.45
MAPK14 Q16539 2/20 0.42
MAPK13 O15264 1/20 0.42
MAPK12 P53778 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825577 0.87 SMYD3 (0.58) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2825617 0.85 TUBB4A (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1518413 0.84 SMYD3 (0.58) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2822965 0.81 SMYD3 (0.52) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2826250 0.80 TUBB4A (0.56) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL12027226 0.78 SMYD3 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2825584 0.78 MAPK14 (0.60) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL2909582 0.78 RAB9A (0.57) SMYD3KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL16236344 0.76 SMYD3 (0.51) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8443948 0.76 PTGS1 (0.40) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069504-A1 (3-OXO)PYRIDIN-4-YLUREA DERIVATIVES AS PDE4 INHIBITORS ALMIRALL, S.A. (ES) 2010-06-24 WO disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed