SCHEMBL28214445

SCHEMBL28214445

N=C(N)NCC(=O)Oc1ccc(I)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
ESR1 P03372 2/20 0.33
HIF1A Q16665 2/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
PRSS1 P07477 4/20 0.33
TMPRSS15 P98073 4/20 0.33
ITGB3 P05106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27257811 0.85 MAPT (0.41) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL27357774 0.85 MAPT (0.41) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL27502925 0.84 MGLL (0.42) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL27532791 0.84 KMT2A (0.43) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL27375786 0.84 LMNA (0.47) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL27182663 0.83 PRSS1 (0.44) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL28174636 0.82 PRSS1 (0.43) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL28199148 0.82 PRSS1 (0.43) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL28249251 0.82 PRSS1 (0.43) KMT2AALDH1A1LMNAMAPTHTT
SCHEMBL28753675 0.81 SMN1; SMN2 (0.47) KMT2AALDH1A1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108698991-A 2-oxoindole compound 凯莫森特里克斯股份有限公司 2018-10-23 CN disclosed
CN-108026050-A NOVEL COMPOUNDS AS ROR GAMMA MODULATORS 格兰马克药品股份有限公司 2018-05-11 CN disclosed
CN-108026039-A New carbocyclic compound as ROR gamma modulators 格兰马克药品股份有限公司 2018-05-11 CN disclosed