Bromide

Bromide

SCHEMBL28214529

Br.Br.Br.Cc1ccccc1C(F)(F)F

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 2/20 0.45
HSD11B1 P28845 5/20 0.45
TSHR P16473 2/20 0.45
TDP1 Q9NUW8 4/20 0.41
ALDH1A1 P00352 3/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AR P10275 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
SCN8A Q9UQD0 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169124 0.97 TSHR (0.47) HSD11B1ACHETSHRTDP1ALDH1A1
SCHEMBL29656610 0.97 TSHR (0.47) HSD11B1ACHETSHRTDP1ALDH1A1
Ammonia Solution, Strong SCHEMBL1870627 0.95 HSD11B1 (0.45) HSD11B1ACHETSHRTDP1ALDH1A1
Hydrochloric Acid SCHEMBL27874688 0.95 TDP1 (0.46) HSD11B1ACHETSHRTDP1ALDH1A1
Fluoride SCHEMBL27976646 0.95 HSD11B1 (0.45) HSD11B1ACHETSHRTDP1ALDH1A1
Acetonitrile SCHEMBL10788322 0.86 AR (0.47) HSD11B1ACHETSHRTDP1ALDH1A1
SCHEMBL11623026 0.81 ACHE (0.47) HSD11B1ACHETSHRTDP1ALDH1A1
SCHEMBL25951815 0.81 ACHE (0.47) HSD11B1ACHETSHRTDP1ALDH1A1
SCHEMBL9568248 0.81 MEN1 (0.43) HSD11B1TSHRTDP1ALDH1A1KDM4E
SCHEMBL10034988 0.79 ACHE (0.45) HSD11B1ACHETSHRTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107954822-A A kind of method for preparing diaryl acetylene compound 浙江大学 2018-04-24 CN disclosed