SCHEMBL28214770

SCHEMBL28214770

CCCCc1ncc2ncn(Cc3ccc(CN)cc3)c2n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.43
TLR7 Q9NYK1 8/20 0.38
TLR8 Q9NR97 3/20 0.38
BRD4 O60885 1/20 0.37
LMNA P02545 2/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC1 Q13547 1/20 0.35
FGFR1 P11362 1/20 0.35
FGFR4 P22455 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
USP1 O94782 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28214165 0.86 MET (0.45) HDAC6TLR7BRD4LMNAHTT
SCHEMBL28214100 0.77 HTT (0.48) LMNAHTTTSHR
SCHEMBL28214711 0.74 YTHDC1 (0.47)
SCHEMBL28214704 0.73 MEN1 (0.42) LMNATSHR
SCHEMBL28214163 0.73 CNR2 (0.43)
SCHEMBL28214101 0.72 CNR2 (0.36) LMNATSHRUSP1
SCHEMBL7491638 0.71 PDE4A (0.58) TLR7
SCHEMBL28214705 0.71 YTHDC1 (0.42) TLR7LMNAHTTTSHRNPSR1
SCHEMBL23764023 0.70 TLR7 (0.46) TLR7TLR8
SCHEMBL6945092 0.69 HDAC6 (0.64) HDAC6LMNAHTTSMN1; SMN2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209466-B purine derivatives as CB2 receptor agonists 豪夫迈·罗氏有限公司 2018-05-18 CN claimed
CN-105209466-B purine derivatives as CB2 receptor agonists 豪夫迈·罗氏有限公司 2018-05-18 CN disclosed