SCHEMBL28215142

SCHEMBL28215142

CC(=O)Oc1ccccc1-c1ncnc(-c2cccs2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMIGD3 P0DMS9 2/20 0.47
ADORA2A P29274 2/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
TSHR P16473 2/20 0.47
GAA P10253 5/20 0.46
LMNA P02545 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 5/20 0.43
NPC1 O15118 4/20 0.43
PDE5A O76074 1/20 0.41
MAPT P10636 6/20 0.40
KDM4E B2RXH2 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
PKM P14618 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
MAOB P27338 1/20 0.39
TP53 P04637 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048688 0.81 TMIGD3 (0.58) TMIGD3ADORA2ASMN1; SMN2TSHRGAA
SCHEMBL27110794 0.74 KDM4E (0.50) SMN1; SMN2GAARAB9ANPC1MAPT
SCHEMBL18938333 0.71 TSHR (0.56) ADORA2ASMN1; SMN2TSHRGAALMNA
SCHEMBL8676653 0.69 PTGS2 (0.61) SMN1; SMN2TSHRGAALMNAALOX15
SCHEMBL28772850 0.69 NPC1 (0.46) ADORA2ASMN1; SMN2GAALMNAMAPK1
SCHEMBL8379241 0.69 TSHR (0.56) TMIGD3ADORA2ASMN1; SMN2TSHRGAA
SCHEMBL20805585 0.67 NPC1 (0.44) ADORA2ASMN1; SMN2GAARAB9ANPC1
SCHEMBL27494568 0.66 TMIGD3 (0.51) TMIGD3ADORA2ASMN1; SMN2TSHRGAA
SCHEMBL27494569 0.66 ADORA2A (0.51) TMIGD3ADORA2ATSHRGAALMNA
SCHEMBL4318402 0.66 ALDH1A1 (0.46) TMIGD3ADORA2ASMN1; SMN2TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108069916-A A kind of 2,4- diaryl for preparing phenyl ring ortho position acetoxylation substitutes the method for -1,3,5 pyrrolotriazine derivatives 中国科学院大连化学物理研究所 2018-05-25 CN disclosed