SCHEMBL28215162

SCHEMBL28215162

CCN(CC)CCc1ccc2ccccc2n1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 6/20 0.49
CYP1A2 P05177 3/20 0.45
CYSLTR1 Q9Y271 2/20 0.45
CYSLTR2 Q9NS75 1/20 0.45
NCF1 P14598 1/20 0.43
GPBAR1 Q8TDU6 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13381947 0.84 HDAC1 (0.48) PDE10ACYP1A2CYSLTR1CYSLTR2NCF1
SCHEMBL27953062 0.84 HDAC1 (0.48) PDE10ACYP1A2CYSLTR1CYSLTR2NCF1
SCHEMBL7749585 0.81 PDE10A (0.51) PDE10ACYP1A2CYSLTR1CYSLTR2NCF1
SCHEMBL725176 0.81 PDE10A (0.54) PDE10ACYP1A2CYSLTR1CYSLTR2GPBAR1
SCHEMBL2913941 0.80 PDE10A (0.61) PDE10ACYP1A2CYSLTR1CYSLTR2NCF1
SCHEMBL29047068 0.79 PDE10A (0.53) PDE10ACYP1A2CYSLTR1CYSLTR2GPBAR1
Iodide SCHEMBL1343671 0.79 PDE10A (0.53) PDE10ACYP1A2CYSLTR1CYSLTR2GPBAR1
SCHEMBL5659096 0.79 PDE10A (0.65) PDE10ACYP1A2CYP2C9PKM
SCHEMBL538491 0.78 GPBAR1 (0.54) PDE10ACYP1A2CYSLTR1CYSLTR2GPBAR1
SCHEMBL6583964 0.77 PDE10A (0.50) PDE10ACYP1A2CYSLTR1CYSLTR2NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108003097-A A kind of synthetic method of cinchocaine 山东诚汇双达药业有限公司 2018-05-08 CN claimed
CN-108003097-A A kind of synthetic method of cinchocaine 山东诚汇双达药业有限公司 2018-05-08 CN disclosed