SCHEMBL2821537

SCHEMBL2821537

Cc1nc2c(C(C)(C)C)cccc2c(-c2ccccc2)c1C(=O)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
ESR1 P03372 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
TACR1 P25103 2/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
PRNP P04156 1/20 0.39
PPARG P37231 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NR2E3 Q9Y5X4 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2821849 0.84 GAA (0.46) GAAMAPTNPSR1NR1H2NR1H3
SCHEMBL2825609 0.81 SMN1; SMN2 (0.44) GAAMAPTNPSR1NR1H2NR1H3
SCHEMBL2821858 0.81 MAPT (0.68) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL1125943 0.81 GAA (0.64) GAAMAPTNPSR1NR1H2NR1H3
SCHEMBL6024428 0.81 ESR1 (0.51) GAAMAPTNPSR1NR1H2NR1H3
SCHEMBL2824028 0.79 FABP3 (0.43) GAAMAPTNPSR1NR1H2NR1H3
SCHEMBL2825677 0.78 FABP3 (0.45) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2821880 0.78 FABP3 (0.45) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2826514 0.77 TACR1 (0.42) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2823196 0.77 GAA (0.40) GAAMAPTNPSR1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed