SCHEMBL2823196

SCHEMBL2823196

Cc1nc2c(N3CC(O)C3)cccc2c(-c2ccccc2)c1C(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
TACR1 P25103 2/20 0.37
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
FABP3 P05413 2/20 0.35
FABP4 P15090 2/20 0.35
PRNP P04156 1/20 0.35
PPARG P37231 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NR2E3 Q9Y5X4 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
ALDH1A1 P00352 2/20 0.34
RBP4 P02753 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2821290 0.92 DGAT1 (0.38) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2824314 0.92 ENPP1 (0.35) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2824028 0.88 FABP3 (0.43) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2821880 0.87 FABP3 (0.45) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2825677 0.87 FABP3 (0.45) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2826514 0.86 TACR1 (0.42) GAAMAPTNPSR1SMN1; SMN2TACR1
SCHEMBL2826068 0.85 NPSR1 (0.43) GAAMAPTNPSR1SMN1; SMN2LMNA
SCHEMBL2824392 0.85 RAF1 (0.37) TACR1ENPP1
SCHEMBL2825178 0.84 CHEK2 (0.41) TACR1
SCHEMBL2828042 0.82 MAPT (0.37) GAAMAPTNPSR1SMN1; SMN2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed